Dab tsi yog qhov txawv ntawm plaub hom "paclitaxel"?

Paclitaxel, tseem hu ua liab paclitaxel, tamsulosin, violet, thiab tesu, yog qhov zoo tshaj plaws natural anti-cancer tshuaj nrhiav pom tam sim no, thiab tau siv dav hauv kev kho mob qog noj ntshav, mob qog noj ntshav, thiab qee cov qog nqaij hlav hauv lub taub hau thiab caj dab thiab. mob ntsws cancer.Raws li cov tshuaj siv tshuaj khomob classical, lub npe ntawmpaclitaxelntseeg tias muaj coob tus neeg tau hnov ​​​​txog nws. Cia peb saib qhov sib txawv ntawm plaub hom paclitaxel hauv kab lus hauv qab no.

paclitaxel

Qhov txawv ntawm plaub hompaclitaxel

1, Paclitaxel: Nws ua rau microtubule / microtubule protein system, inhibits microtubule depolymerization, thaiv lub voj voog ntawm tes hauv G2 / M theem, ua rau mitosis txawv txav lossis raug ntes, tiv thaiv qog cell replication, thiab ua rau cov qog nqaij hlav tsis tuaj yeem mus txuas ntxiv thiab tuag.

2, Docetaxel: Cov txheej txheem ntawm kev ua haujlwm yog tib yam li ntawm paclitaxel, tab sis nrog ntau dua affinity rau microtubule khi qhov chaw thiab ntau dua kev tiv thaiv kab mob.

3, Liposomal paclitaxel: Cov txheej txheem ntawm kev ua haujlwm yog tib yam li ntawm paclitaxel.Cov liposomes muaj lecithin, cholesterol, threonine thiab lwm yam ntaub ntawv zoo ib yam li phospholipid bilayer qauv ntawm cell membranes encapsulate paclitaxel, uas tuaj yeem txhim kho cov dej solubility, nkag tau yooj yim dua. rau hauv cov qog nqaij hlav los ntawm cov hlab ntsha, thiab txo cov toxicity ntawm lub plawv thiab lub raum, thiab lwm yam.

4.Albumin-bound paclitaxel: hydrophobic paclitaxel yog ua ke nrog tib neeg cov ntshav albumin cab kuj los ntawm nanotechnology.Albumin tuaj yeem ua rau kom cov paclitaxel nyob rau hauv cov qog los ntawm kev khi rau gp60 receptor thiab nce qhov concentration ntawm paclitaxel hauv cov ntaub so ntswg, yog li ua rau cov nyhuv tiv thaiv qog. .

Ob leeg paclitaxel, doxorubicin, paclitaxel liposome los yog albumin paclitaxel yog tib hom tshuaj chemotherapeutic, thiab tag nrho cov nyob rau hauv cov chav kawm ntawm paclitaxel nyob rau hauv kev faib cov tshuaj chemotherapeutic.Lawv yog tib hom tshuaj.Paclitaxel yog ib qho tshuaj antitumor nrog lub hauv paus ntsiab lus ntawm microtubule. inhibitor, uas yog siv dav hauv kev kho mob qog noj ntshav mis.

Nco tseg: Cov kev ua tau zoo thiab cov ntawv thov hauv qhov kev nthuav qhia no yog muab los ntawm cov ntaub ntawv luam tawm.

Paclitaxel API

Kev nyeem ntawv txuas ntxiv:Yunnan Hande Biotechnology Co., Ltd. tau tsom mus rau kev tsim cov paclitaxel rau 28 xyoo.Nws yog lub ntiaj teb thawj tus neeg ua haujlwm ywj pheej ntawm cov nroj tsuag-derived anticancer tshuaj paclitaxel uas tau pom zoo los ntawm US FDA, European EDQM, Australian TGA, Tuam Tshoj CFDA, Is Nrias teb, Nyiv thiab lwm lub tebchaws tswj hwm.kev lag luam.Yog xav yuavPaclitaxel API, thov hu rau peb hauv online.


Post lub sij hawm: Oct-08-2022